{737789-87-6 relugolix
CAS: 737789-87-6
MF: C29H27F2N7O5S
MW: 623.63
Einecs: 237-099-7
MDL No.:MFCD25976856
Airíonna
Cuma bán ar sholad criostalach as-bán
Leáphointe: 228 céim (decomp)
Dlús 1.442 ± 0. 06 g/cm3
Teocht stórála. Stóráil ag céim -20
Intuaslagthacht DMSO: 2 0. 0 (Max Conc. mg/ml);
Eatánól: 1. 0 (max conc. Mg/ml);
Iarratas:
Is freasúra GNRH é Relugolix, ar a dtugtar freasúra gabhdóra hormóin a scaoileann gonadotropin freisin. Murab ionann agus an chuid is mó de na modhnaitheoirí GnRH eile, ach cosúil le Elalagolix (ainm trádála orilissa), is comhdhúil mhóilíneach beag neamh -peiptíde é Relugolix is féidir a thógáil ó bhéal. Féadann sé leibhéil hormóin ghnéas fireann agus baineann a chosc go dtí an raon iar -mhíostraithe nó an ration.
Comhchiallaigh:
Relugolix
737789-87-6
Tak -385
Orgovyx
Tak 385
{1- ({4- ({1- (2, 6- difluOrobenzyl) -5- (((dimethylamino) methyl) -3- ({{{{}}} methoxypyrazin {8}} ({{{}}} methoxypyrazin {8}} yl) {-2, {4- déxo {-1, 2,3, {4- tetrahydrothieno [2, 3- d] pyrimidin -6- yl) phenyl) {{{18} methoxyurea)
Relugolix comhpháirt myfembree
{1- [4- [{1- [(2, 6- difluorophenyl) methyl] -5- [(dimethylamino) methyl] ypyridazin {-3- yl) {-2, {4- déxothieno [2, 3- d] pyrimidin {-6- yl] feinil] -3- methoxyurea
N-({4- ({1- ((2, {{}}} difluorophenyl) methyl) -5- ((dimethylamino) methyl) -1, 2,3, {{{4- tetrahydo {}} (}} ({4- tetrahyDDO}}}}}}}} tetrahyDDO}}}} tetrahyd {6- methoxy {-3- pyridazinyl) {-2, {4- déxothieno (2, 3- d) pyrimidin -6- yl) -n'-mothoxyurea)
Úiré, N-({4- ({1- ((2, {{}}} difluorophenyl) methyl) -5- ((dimethylamino) methyl) -1, 2,3, {{{4- tetrahyDDO {}}}}}}} .
Relugolix
Relugolixum
Tak385
{1- ({4- ({1- ((2, 6- difluorophenyl) -5- ((dimethylamino) methyl) -3- ({6- methoxyPyridin -3- (6-}}} {}}}}}}}}}}}}}}}}}}}}}}}} {{{}}} ({{}}}} } Yl) -2, {4- déxo {-1, 2,3, {4- tetrahydrothieno (2, {3- d) pyrimidin -6-} yl) {
{1- (4- {{1- [(2, 6- difluorophenyl) methyl] -5- [(dimethylamino) methyl] {{{}} ({6- {}} methoxyRidin {8}} ({{}}}}}} {}}}}}}}}}}}} { } yl) -2, {4- déxo {-1, 2,3, {4- tetrahydrothieno [2, 3- d] pyrimidin -6-} yl}}}}}}}}}}}}}}}}}}}}}}}}}}}}}
Orgovyx
Clibeanna Te: {737789-87-6 relugolix, an tSín 737789-87-6 Déantúsóirí, soláthróirí


